Bitopic Ligands and Metastable Binding Sites: Opportunities for G Protein-Coupled Receptor (GPCR) Medicinal Chemistry-Reference-Cited by-同舟云学术

Bitopic Ligands and Metastable Binding Sites: Opportunities for G Protein-Coupled Receptor (GPCR) Medicinal Chemistry

Published:2017-02-15 Issue:10 Volume:60 Page:4126-4134
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fronik Philipp¹,Gaiser Birgit I.¹,Sejer Pedersen Daniel¹^ORCID

Affiliation:

1. Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Jagtvej 162, 2100 Copenhagen, Denmark

Funder

Carlsbergfondet

Det Sundhedsvidenskabelige Fakultet, K?benhavns Universitet

Lundbeckfonden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b01601

Reference93 articles.

1. The GPCR Network: a large-scale collaboration to determine human GPCR structure and function

2. The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints

3. Structure-Function of the G Protein–Coupled Receptor Superfamily

4. Structural diversity of G protein-coupled receptors and significance for drug discovery

5. How many drug targets are there?

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