The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold-Reference-Cited by-同舟云学术

The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold

Published:2017-08-14 Issue:16 Volume:60 Page:6880-6896
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sandoval Elena¹,Lafuente-Monasterio María José¹,Almela María J.¹,Castañeda Pablo¹,Jiménez Díaz María Belén¹,Martínez-Martínez María S.¹,Vidal Jaume¹,Angulo-Barturen Íñigo¹,Bamborough Paul²,Burrows Jeremy³,Cammack Nicholas¹,Chaparro María J.¹,Coterón José M.¹,de Cozar Cristina¹,Crespo Benigno¹,Díaz Beatriz¹,Drewes Gerard⁴,Fernández Esther¹,Ferrer-Bazaga Santiago¹,Fraile María Teresa¹,Gamo Francisco J.¹,Ghidelli-Disse Sonja⁴,Gómez Rubén¹,Haselden John¹,Huss Sophie¹,León María Luisa¹,de Mercado Jaime¹,Macdonald Simon J. F.²^ORCID,Martín Hernando José Ignacio¹,Prats Sara¹,Puente Margarita¹,Rodríguez Anne¹,de la Rosa Juan C.¹,Rueda Lourdes¹,Selenski Carolyn⁵,Willis Paul³,Wilson David M.¹,Witty Michael³,Calderón Félix¹^ORCID

Affiliation:

1. Tres Cantos, Medicines Development Campus, DDW, GlaxoSmithKline, Severo Ochoa 2, 28760 Tres Cantos, Madrid, Spain

2. Medicines Research Center, GlaxoSmithKline, Gunnels Wood Road, Stevenage SG1 2NY, U.K.

3. Medicines for Malaria Venture (MMV), 21 route de Pré-Bois, PO Box 1826, 1215 Geneva 15, Switzerland

4. Cellzome GmbH, GlaxoSmithKline, Meyerhofstrasse 1, 69117 Heidelberg, Germany

5. GlaxoSmithKline, 709 Swedeland Road, King of Prussia, Pennsylvania 19406, United States

Funder

Medicines for Malaria Venture

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b01441

Reference35 articles.

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3. The economic and social burden of malaria

4. Trends in Reported Malaria Incidence;World Health Organization:Geneva, 2016; http://www.who.int/en/(accessed Nov 19, 2016).

5. Pyrethroid resistance in African anopheline mosquitoes: what are the implications for malaria control?

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