Synthesis and in Vivo Biological Evaluation of 68Ga-Labeled Carbonic Anhydrase IX Targeting Small Molecules for Positron Emission Tomography

Author:

Sneddon Deborah1,Niemans Raymon2,Bauwens Matthias3,Yaromina Ala2,van Kuijk Simon J. A.2,Lieuwes Natasja G.2,Biemans Rianne2,Pooters Ivo3,Pellegrini Paul A.4,Lengkeek Nigel A.4,Greguric Ivan4,Tonissen Kathryn F.1,Supuran Claudiu T.5,Lambin Philippe2,Dubois Ludwig2,Poulsen Sally-Ann1

Affiliation:

1. Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland 4111, Australia

2. Maastricht Radiation Oncology (MAASTRO Lab), GROW − School for Oncology and Developmental Biology, Maastricht University, Medical Centre, 6200 MD Maastricht, The Netherlands

3. Departments of Radiology and Nuclear Medicine, Maastricht University Medical Centre, 6202 AZ Maastricht, The Netherlands

4. LifeSciences Division, Australian Nuclear Science and Technology Organisation (ANSTO), Locked Bag 2001, Kirrawee DC, New South Wales 2232, Australia

5. Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche, Polo Scientifico, Università degli Studi di Firenze, 50019 Sesto Fiorentino, Italy

Funder

Australian Research Council

Australian Institute of Nuclear Science and Engineering

KWF Kankerbestrijding

Cancer Council Queensland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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