Identification of the Binding Site of Chroman-4-one-Based Sirtuin 2-Selective Inhibitors using Photoaffinity Labeling in Combination with Tandem Mass Spectrometry-Reference-Cited by-同舟云学术

Identification of the Binding Site of Chroman-4-one-Based Sirtuin 2-Selective Inhibitors using Photoaffinity Labeling in Combination with Tandem Mass Spectrometry

Published:2016-11-21 Issue:23 Volume:59 Page:10794-10799
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Seifert Tina¹,Malo Marcus¹,Lengqvist Johan²,Sihlbom Carina²,Jarho Elina M.³,Luthman Kristina¹

Affiliation:

1. Department of Chemistry and Molecular Biology, Medicinal Chemistry, University of Gothenburg, Kemivagen 10, SE-41296 Göteborg, Sweden

2. The Proteomics Core Facility, Sahlgrenska Academy, University of Gothenburg, SE-41390 Göteborg, Sweden

3. School of Pharmacy, University of Eastern Finland, P.O. Box 1627, 70211 Kuopio, Finland

Funder

Vetenskapsrådet

European Cooperation in Science and Technology

Göteborgs Universitet

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b01117

Reference28 articles.

1. Photoaffinity labeling in target- and binding-site identification

2. Photoaffinity Labeling in Drug Discovery and Developments: Chemical Gateway for Entering Proteomic Frontier

3. Development and application of diazirines in biological and synthetic macromolecular systems

4. A propofol binding site on mammalian GABAA receptors identified by photolabeling

5. Photoaffinity Labeling of Nicotinic Receptors: Diversity of Drug Binding Sites!

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