Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine Derivatives: New Highly Potent A2A Adenosine Receptor Inverse Agonists with Antinociceptive Activity-Reference-Cited by-同舟云学术

Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine Derivatives: New Highly Potent A2A Adenosine Receptor Inverse Agonists with Antinociceptive Activity

Published:2016-11-29 Issue:23 Volume:59 Page:10564-10576
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Varano Flavia¹,Catarzi Daniela¹,Vincenzi Fabrizio²,Betti Marco¹,Falsini Matteo¹,Ravani Annalisa²,Borea Pier Andrea²,Colotta Vittoria¹,Varani Katia²

Affiliation:

1. Dipartimento di Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino, Sezione di Farmaceutica e Nutraceutica, Università degli Studi di Firenze, via Ugo Schiff, 6, 50019, Sesto Fiorentino, Italy

2. Dipartimento di Scienze Mediche, Sezione di Farmacologia, Università degli Studi di Ferrara, via Fossato di Mortara 17-19, 44121, Ferrara, Italy

Funder

Ministero dell’Istruzione, dell’Università e della Ricerca

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b01068

Reference59 articles.

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