Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity

Author:

Travelli Cristina1,Aprile Silvio1,Rahimian Reza23,Grolla Ambra A.1,Rogati Federica1,Bertolotti Mattia1,Malagnino Floriana1,di Paola Rosanna4,Impellizzeri Daniela4,Fusco Roberta4,Mercalli Valentina1,Massarotti Alberto1ORCID,Stortini Giorgio5,Terrazzino Salvatore1,Del Grosso Erika1,Fakhfouri Gohar2,Troiani Maria Pia6,Alisi Maria Alessandra6,Grosa Giorgio1,Sorba Giovanni1,Canonico Pier Luigi1,Orsomando Giuseppe7,Cuzzocrea Salvatore4,Genazzani Armando A.1,Galli Ubaldina1ORCID,Tron Gian Cesare1

Affiliation:

1. Dipartimento di Scienze del Farmaco, Università degli Studi del Piemonte Orientale “A. Avogadro”, Largo Donegani 2, 28100 Novara, Italy

2. Department of Pharmacology, School of Medicine, Tehran University of Medical Sciences, Tehran, Iran

3. Department of Psychiatry and Neuroscience, Faculty of Medicine, Research Center of the Mental Health Institute of Quebec, Laval University, Quebec, Quebec G1J 2G3, Canada

4. Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, Via C. Valeria Gazzi, 98100 Messina, Italy

5. Department of Oncology, Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano, Milan, Italy

6. R&D, Angelini Research Center, Piazzale della Stazione, 00040 S. Palomba-Pomezia, Italy

7. Department of Clinical Sciences (DISCO), Section of Biochemistry, Polytechnic University of Marche, Via Ranieri 67, 60131 Ancona, Italy

Funder

Ministero dell?Istruzione, dell?Universit? e della Ricerca

Associazione Italiana per la Ricerca sul Cancro

Universit? degli Studi del Piemonte Orientale

Fondazione San Paolo

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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