Identification and SAR Evaluation of Hemozoin-Inhibiting Benzamides Active against Plasmodium falciparum-Reference-Cited by-同舟云学术

Identification and SAR Evaluation of Hemozoin-Inhibiting Benzamides Active against Plasmodium falciparum

Published:2016-06-24 Issue:13 Volume:59 Page:6512-6530
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wicht Kathryn J.¹,Combrinck Jill M.¹²,Smith Peter J.²,Hunter Roger¹,Egan Timothy J.¹

Affiliation:

1. Department of Chemistry, University of Cape Town, Rondebosch 7701, South Africa

2. Division of Pharmacology, Department of Medicine, Faculty of Health Sciences, University of Cape Town, Observatory 7925, South Africa

Funder

National Institute of Allergy and Infectious Diseases

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6b00719

Reference86 articles.

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2. That Was Then But This Is Now: Malaria Research in the Time of an Eradication Agenda

3. Genomic Insights into the Past, Current and Future Evolution of Human Parasites of the Genus Plasmodium

4. Studies of resistance to chloroquine, quinine, amodiaquine and mefloquine among Philippine strains of Plasmodium falciparum

5. Selection for mefloquine resistance in Plasmodium falciparum is linked to amplification of the pfmdr1 gene and cross-resistance to halofantrine and quinine.

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