A Small-Molecule Oral Agonist of the Human Glucagon-like Peptide-1 Receptor
Author:
Affiliation:
1. Pfizer Worldwide Research, Development, and Medical, Cambridge, Massachusetts 02139, United States
2. Pfizer Worldwide Research, Development, and Medical, Groton, Connecticut 06340, United States
3. Sosei Heptares, Cambridge CB21 6DG, U.K.
Funder
Pfizer
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01856
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3. Tissue and Plasma Concentrations of Amidated and Glycine-Extended Glucagon-Like Peptide I in Humans
4. GLUCAGON-LIKE PEPTIDE-1 7-36: A PHYSIOLOGICAL INCRETIN IN MAN
5. Glucagon-like peptide 1 inhibition of gastric emptying outweighs its insulinotropic effects in healthy humans
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