Target Fishing Reveals a Novel Mechanism of 1,2,4-Oxadiazole Derivatives Targeting Rpn6, a Subunit of 26S Proteasome-Reference-Cited by-同舟云学术

Target Fishing Reveals a Novel Mechanism of 1,2,4-Oxadiazole Derivatives Targeting Rpn6, a Subunit of 26S Proteasome

Published:2022-03-06 Issue:6 Volume:65 Page:5029-5043
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Dai Zhen¹²,An Lu-yan¹²,Chen Xiao-yi¹²,Yang Fan¹²,Zhao Ni¹²,Li Cui-cui¹²,Ren Ren¹²,Li Bing-yan¹²,Tao Wei-yan¹²,Li Pei¹²,Jiang Cheng¹²,Yan Fang¹²,Jiang Zheng-yu¹,You Qi-dong¹^ORCID,Di Bin¹²^ORCID,Xu Li-li¹²^ORCID

Affiliation:

1. Jiangsu Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China

2. Key Laboratory of Drug Quality Control and Pharmacovigilance, Ministry of Education, China Pharmaceutical University, Nanjing 210009, China

Funder

Ministry of Science and Technology of the People's Republic of China

China Pharmaceutical University

Natural Science Foundation of Jiangsu Province

Central University Basic Research Fund of China

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c02210

Reference85 articles.

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