Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe-Reference-Cited by-同舟云学术

Development of a Selective Dual Discoidin Domain Receptor (DDR)/p38 Kinase Chemical Probe

Published:2021-09-10 Issue:18 Volume:64 Page:13451-13474
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Röhm Sandra¹²^ORCID,Berger Benedict-Tilman¹²^ORCID,Schröder Martin¹²^ORCID,Chatterjee Deep¹²,Mathea Sebastian¹²^ORCID,Joerger Andreas C.¹²^ORCID,Pinkas Daniel M.³^ORCID,Bufton Joshua C.³,Tjaden Amelie¹²,Kovooru Lohitesh²⁴,Kudolo Mark⁵,Pohl Christian²⁴,Bullock Alex N.³^ORCID,Müller Susanne¹²^ORCID,Laufer Stefan⁵^ORCID,Knapp Stefan¹²^ORCID

Affiliation:

1. Institute of Pharmaceutical Chemistry, Johann Wolfgang Goethe University, Max-von-Laue-Str. 9, 60438 Frankfurt am Main, Germany

2. Structural Genomics Consortium (SGC), Buchmann Institute for Molecular Life Sciences, Max-von-Laue-Str. 15, 60438 Frankfurt am Main, Germany

3. Centre for Medicines Discovery, University of Oxford, Old Road Campus, Roosevelt Drive, Oxford OX3 7DQ, U.K.

4. Institute of Biochemistry II, Faculty of Medicine, Johann Wolfgang Goethe University, Max-von-Laue-Str. 15, 60438 Frankfurt am Main, Germany

5. Department of Pharmaceutical/Medicinal Chemistry, Eberhard Karls University Tübingen, Auf der Morgenstelle 8, 72076 Tübingen, Germany

Funder

H2020 Research Infrastructures

Structural Genomics Consortium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00868

Reference42 articles.

1. An Orphan Receptor Tyrosine Kinase Family Whose Members Serve as Nonintegrin Collagen Receptors

2. The Discoidin Domain Receptor Tyrosine Kinases Are Activated by Collagen

3. Small Molecule Discoidin Domain Receptor Kinase Inhibitors and Potential Medical Applications

4. Molecular Analysis of Collagen Binding by the Human Discoidin Domain Receptors, DDR1 and DDR2

5. Discoidin domain receptors: Micro insights into macro assemblies

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