Selective Penicillamine Substitution Enables Development of a Potent Analgesic Peptide that Acts through a Non-Opioid-Based Mechanism-Reference-Cited by-同舟云学术

Selective Penicillamine Substitution Enables Development of a Potent Analgesic Peptide that Acts through a Non-Opioid-Based Mechanism

Published:2021-06-18 Issue:13 Volume:64 Page:9271-9278
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gajewiak Joanna¹^ORCID,Christensen Sean B.¹,Dowell Cheryl¹,Hararah Fuaad¹,Fisher Fernando¹,Huynh Peter N.¹,Olivera Baldomero M.¹,McIntosh J. Michael¹²³

Affiliation:

1. School of Biological Sciences, University of Utah, 257 South 1400 East, Salt Lake City, Utah 84112-0840, United States

2. George E. Wahlen Department of Veterans Affairs Medical Center, 500 Foothill Dr., Salt Lake City, Utah 84148, United States

3. Department of Psychiatry, University of Utah, 501 Chipeta Way, Salt Lake City, Utah 84108, United States

Funder

National Institute of General Medical Sciences

Office of the Assistant Secretary of Defense for Health Affairs

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00512

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5. Therapeutic applications of conotoxins that target the neuronal nicotinic acetylcholine receptor

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