Discovery of a Potent FLT3 Inhibitor (LT-850-166) with the Capacity of Overcoming a Variety of FLT3 Mutations

Author:

Wang Zhijie1,Cai Jiongheng1,Ren Jiwei1,Chen Yun2,Wu Yingli3,Cheng Jie1,Jia Kun1,Huang Fei1,Cheng Zitian1,Sheng Tiancheng4,Song Shiyu5,Heng Hao6,Zhu Yifan7,Tang Weifang1ORCID,Li Hongmei1,Lu Tao8,Chen Yadong9ORCID,Lu Shuai1ORCID

Affiliation:

1. School of Science, China Pharmaceutical University, Nanjing 211198, P. R. China

2. Edmond H. Fischer Translational Medical Research Laboratory, Scientific Research Center, The Seventh Affiliated Hospital, Sun Yat-Sen University, Shenzhen 518107, P. R. China

3. Chemical Biology Division of Shanghai Universities E-Institutes, Hongqiao International Institute of Medicine, Shanghai Tongren Hospital/Faculty of Basic Medicine, Key Laboratory of Cell Differentiation and Apoptosis of the Chinese Ministry of Education, Shanghai Jiao Tong University School of Medicine, Shanghai 200025, P. R. China

4. School of Engineering, China Pharmaceutical University, Nanjing 211198, P. R. China

5. School of Life Sciences and Technology, China Pharmaceutical University, Nanjing 210038, P. R. China

6. Department of Polymer Science & Engineering, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210023, P. R. China

7. School of Pharmacy, China Pharmaceutical University, Nanjing 210009, P.R. China

8. State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing 210009, P. R. China

9. Laboratory of Molecular Design and Drug Discovery, China Pharmaceutical University, Nanjing 211198, P. R. China

Funder

China Pharmaceutical University

Natural Science Foundation of Jiangsu Province

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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