Discovery of 5-{2-[5-Chloro-2-(5-ethoxyquinoline-8-sulfonamido)phenyl]ethynyl}-4-methoxypyridine-2-carboxylic Acid, a Highly Selective in Vivo Useable Chemical Probe to Dissect MCT4 Biology-Reference-Cited by-同舟云学术

Discovery of 5-{2-[5-Chloro-2-(5-ethoxyquinoline-8-sulfonamido)phenyl]ethynyl}-4-methoxypyridine-2-carboxylic Acid, a Highly Selective in Vivo Useable Chemical Probe to Dissect MCT4 Biology

Published:2021-08-12 Issue:16 Volume:64 Page:11904-11933
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Heinrich Timo¹^ORCID,Sala-Hojman Ada¹,Ferretti Roberta²,Petersson Carl¹,Minguzzi Stefano³,Gondela Andrzej⁴,Ramaswamy Shivapriya²,Bartosik Anna⁴,Czauderna Frank²,Crowley Lindsey²,Wahra Pamela²,Schilke Heike¹,Böpple Pia¹,Dudek Łukasz⁴,Leś Marcin⁴,Niedziejko Paulina⁴,Olech Kamila⁴,Pawlik Henryk⁴,Włoszczak Łukasz⁴,Zuchowicz Karol⁴,Suarez Alvarez Jose Ramon⁴,Martyka Justyna⁴,Sitek Ewa⁴,Mikulski Maciej⁴,Szczęśniak Joanna⁴,Jäckel Sven¹,Krier Mireille¹^ORCID,Król Marcin⁴,Wegener Ansgar¹,Gałęzowski Michał⁴,Nowak Mateusz⁴,Becker Frank³,Herhaus Christian¹

Affiliation:

1. Merck Healthcare KGaA, Frankfurter Str. 250, 64293 Darmstadt, Germany

2. EMD Serono Research & Development Institute, Inc., 45A Middlesex Turnpike, Billerica, Massachusetts 01821, United States

3. Intana, Bioscience GmbH, Lochhamer Str. 29a, 82152 Planegg, Martinsried, Germany

4. Ryvu Therapeutics, Sternbacha 2, 30-394 Kraków, Poland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00448

Reference36 articles.