Synthesis, Optimization, and Biological Evaluation of Corrinated Conjugates of the GLP-1R Agonist Exendin-4-Reference-Cited by-同舟云学术

Synthesis, Optimization, and Biological Evaluation of Corrinated Conjugates of the GLP-1R Agonist Exendin-4

Published:2021-03-06 Issue:6 Volume:64 Page:3479-3492
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tinsley Ian C.¹,Borner Tito²,Swanson MacKenzie L.¹,Chepurny Oleg G.³,Doebley Sarah A.²,Kamat Varun⁴,Sweet Ian R.⁴,Holz George G.³,Hayes Matthew R.⁵,De Jonghe Bart C.²,Doyle Robert P.¹³^ORCID

Affiliation:

1. Department of Chemistry, Syracuse University, 111 College Place, Syracuse, New York 13244, United States

2. Department of Biobehavioral Health Sciences, University of Pennsylvania, School of Nursing, Philadelphia, Pennsylvania 19104, United States

3. Department of Medicine, State University of New York, Upstate Medical University, Syracuse, New York 13210, United States

4. Department of Medicine, University of Washington, Medicine Diabetes Institute, Seattle, Washington 98109, United States

5. Department of Psychiatry, University of Pennsylvania, Perelman School of Medicine, Philadelphia, Pennsylvania 19104, United States

Funder

Schweizerischer Nationalfonds zur F??rderung der Wissenschaftlichen Forschung

U.S. Department of Health and Human Services

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00185

Reference72 articles.

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