Structure–Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor γt-Reference-Cited by-同舟云学术

Structure–Activity Relationship Studies of Trisubstituted Isoxazoles as Selective Allosteric Ligands for the Retinoic-Acid-Receptor-Related Orphan Receptor γt

Published:2021-05-19 Issue:13 Volume:64 Page:9238-9258
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Meijer Femke A.¹^ORCID,Saris Annet O.W.M.¹,Doveston Richard G.¹²,Oerlemans Guido J.M.¹^ORCID,de Vries Rens M.J.M.¹,Somsen Bente A.¹,Unger Anke³,Klebl Bert³,Ottmann Christian¹^ORCID,Cossar Peter J.¹,Brunsveld Luc¹^ORCID

Affiliation:

1. Laboratory of Chemical Biology, Department of Biomedical Engineering and Institute for Complex Molecular Systems, Technische Universiteit Eindhoven, Den Dolech 2, 5612 AZ Eindhoven, The Netherlands

2. Leicester Institute of Structural and Chemical Biology and School of Chemistry, University of Leicester, University Road, LE1 7RH Leicester, U.K.

3. Lead Discovery Center GmbH, 44227 Dortmund, Germany

Funder

Horizon 2020 Framework Programme

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00475

Reference50 articles.