Thieno[2,3-d]pyrimidine-Based Positive Allosteric Modulators of Human Mas-Related G Protein-Coupled Receptor X1 (MRGPRX1)
Author:
Affiliation:
1. Tsukuba Research Laboratories, Eisai Co., Ltd., Tsukuba, Ibaraki 300-2635, Japan
Funder
National Center for Advancing Translational Sciences
National Institute of Neurological Disorders and Stroke
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01709
Reference16 articles.
1. A Diverse Family of GPCRs Expressed in Specific Subsets of Nociceptive Sensory Neurons
2. Proenkephalin A gene products activate a new family of sensory neuron–specific GPCRs
3. Modulation of Ion Channels and Synaptic Transmission by a Human Sensory Neuron-Specific G-Protein-Coupled Receptor, SNSR4/mrgX1, Heterologously Expressed in Cultured Rat Neurons
4. Activation of MrgC receptor inhibits N-type calcium channels in small-diameter primary sensory neurons in mice
5. TRPA1 is required for histamine-independent, Mas-related G protein–coupled receptor–mediated itch
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