Does the Number of Bifunctional Chelators Conjugated to a mAb Affect the Biological Activity of Its Radio-Labeled Counterpart? Discussion Using the Example of mAb against CD-20 Labeled with <sup>90</sup>Y or <sup>177</sup>Lu-Reference-Cited by-同舟云学术

Does the Number of Bifunctional Chelators Conjugated to a mAb Affect the Biological Activity of Its Radio-Labeled Counterpart? Discussion Using the Example of mAb against CD-20 Labeled with ⁹⁰Y or ¹⁷⁷Lu

Published:2022-04-20 Issue:9 Volume:65 Page:6419-6430
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Karczmarczyk Urszula¹^ORCID,Sawicka Agnieszka¹,Garnuszek Piotr¹,Maurin Michał¹,Wojdowska Wioletta¹

Affiliation:

1. National Centre for Nuclear Research, Radioisotope Centre POLATOM, Otwock 05-400, Poland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c02044

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