Lead Optimization of Influenza Virus RNA Polymerase Inhibitors Targeting PA–PB1 Interaction

Author:

Mizuta Satoshi1ORCID,Otaki Hiroki1ORCID,Ishikawa Takeshi2ORCID,Makau Juliann Nzembi3,Yamaguchi Tomoko1,Fujimoto Takuya4,Takakura Nobuyuki4,Sakauchi Nobuki4,Kitamura Shuji4,Nono Hikaru5,Nishi Ryota5,Tanaka Yoshimasa6,Takeda Kohsuke7,Nishida Noriyuki8,Watanabe Ken9

Affiliation:

1. Center for Bioinformatics and Molecular Medicine, Graduate School of Biomedical Sciences, Nagasaki University, 1-14 Bunkyo, Nagasaki 852-8521, Japan

2. Department of Chemistry, Biotechnology, and Chemical Engineering, Graduate School of Science and Engineering, Kagoshima University, 1-21-40 Korimoto, Kagoshima 890-0065, Japan

3. Center for Virus Research, Kenya Medical Research Institute, 54840-00200 Nairobi, Kenya

4. Chemistry, Discovery Science, Axcelead Drug Discovery Partners, Inc., 26-1, Muraoka-Higashi 2-chome, Fujisawa, Kanagawa 251-0012, Japan

5. School of Medicine, Nagasaki University, 1-12-4 Sakamoto, Nagasaki 852-8523, Japan

6. Center for Medical Innovation, Nagasaki University, 1-7-1 Sakamoto, Nagasaki 852-8588, Japan

7. Department of Cell Regulation, Graduate School of Biomedical Sciences, Nagasaki University, 1-14 Bunkyo, Nagasaki 852-8521, Japan

8. Department of Molecular Microbiology and Immunology, Graduate School of Biomedical Sciences, Nagasaki University, 1-12-4 Sakamoto, Nagasaki 852-8523, Japan

9. Department of Lifestyle Design, Faculty of Human Ecology, Yasuda Women’s University, 6-13-1 Yasuhigashi, Asaminami Ward, Hiroshima 731-0153, Japan

Funder

Japan Agency for Medical Research and Development

Japan Society for the Promotion of Science

Center for Clinical and Translational Research of Kyushu University Hospital

GSK Japan Research Grant 2019

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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