Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy

Author:

Zhang Zhuqing12,Guo Zuhao32,Xu Xiaowei12,Cao Danyan3,Yang Hong1,Li Yanlian3,Shi Qiongyu1,Du Zhiyan3,Guo Xiaobin1,Wang Xin3,Chen Danqi3,Zhang Ying12,Chen Lin3,Zhou Kaixin3,Li Jian4,Geng Meiyu125,Huang Xun125,Xiong Bing32ORCID

Affiliation:

1. Division of Anti-tumor Pharmacology, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, P. R. China

2. University of Chinese Academy of Sciences, NO.19A Yuquan Road, Beijing 100049, P. R. China

3. Department of Medicinal Chemistry, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, P. R. China

4. College of Pharmaceutical Sciences, Gannan Medical University, Ganzhou 341000, P. R. China

5. Hangzhou Institute for Advanced Study, UCAS, Hangzhou 310024, P. R. China

Funder

Shanghai Institutes for Biological Sciences, Chinese Academy of Sciences

American Heart Association

Georgia Cancer Coalition

Science and Technology Commission of Shanghai Municipality

National Natural Science Foundation of China

Georgia State University

State Key Laboratory of Drug Research

Jiangxi "Double Thousand Plan"

Shanghai Municipal Commission of Health and Family Planning

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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