Structure–Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists-Reference-Cited by-同舟云学术

Structure–Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

Published:2021-06-28 Issue:13 Volume:64 Page:9330-9353
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sedlák David¹^ORCID,Wilson Tyler A.²,Tjarks Werner³,Radomska Hanna S.⁴,Wang Hongyan⁴,Kolla Jayaprakash Narayana¹,Leśnikowski Zbigniew J.⁵^ORCID,Špičáková Alena⁶,Ali Tehane³,Ishita Keisuke³,Rakotondraibe Liva Harinantenaina³^ORCID,Vibhute Sandip²,Wang Dasheng²,Anzenbacher Pavel⁶,Bennett Chad²⁷,Bartunek Petr¹,Coss Christopher C.⁴⁷^ORCID

Affiliation:

1. CZ-OPENSCREEN, Institute of Molecular Genetics of the Czech Academy of Sciences, Vídeňská 1083, 142 20 Prague, Czech Republic

2. Medicinal Chemistry Shared Resource, Comprehensive Cancer Center, The Ohio State University, Columbus, Ohio 43210, United States

3. Division of Medicinal Chemistry and Pharmacognosy College of Pharmacy, The Ohio State University, Columbus, Ohio 43210, United States

4. Division of Pharmaceutics and Pharmacology, College of Pharmacy, The Ohio State University, Columbus, Ohio 43210, United States

5. Laboratory of Medicinal Chemistry, Institute of Medical Biology PAS, 106 Lodowa Street, 93-232 Lodz, Poland

6. Department of Pharmacology, Faculty of Medicine, Palacky University, Hněvotínská 3, 77515 Olomouc, Czech Republic

7. Drug Development Institute, Comprehensive Cancer Center, The Ohio State University, Columbus, Ohio 43210, United States

Funder

U.S. Department of Health and Human Services

Ministerstvo ??kolstv??, Ml??de??e a Telov??chovy

Instytut Biologii Medycznej Polskiej Akademii Nauk

Univerzita Palack??ho v Olomouci

Institute of Molecular Genetics of the Czech Academy of Sciences

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c00555

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4. Mechanisms of Estrogen Action

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