One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes-Reference-Cited by-同舟云学术

One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes

Published:2021-12-27 Issue:1 Volume:65 Page:824-837
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Vannozzi Gioele¹,Vullo Daniela¹,Angeli Andrea¹^ORCID,Ferraroni Marta²^ORCID,Combs Jacob³,Lomelino Carrie³,Andring Jacob³^ORCID,Mckenna Robert³,Bartolucci Gianluca¹^ORCID,Pallecchi Marco¹,Lucarini Laura⁴,Sgambellone Silvia⁴,Masini Emanuela⁴,Carta Fabrizio¹^ORCID,Supuran Claudiu T.¹^ORCID

Affiliation:

1. NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, Via Ugo Schiff 6, Sesto Fiorentino, 50019 Florence, Italy

2. Dipartimento di Chimica “ Ugo Schiff”, University of Florence, Via della Lastruccia 3, Sesto Fiorentino, 50019 Florence, Italy

3. Department of Biochemistry and Molecular Biology, College of Medicine, University of Florida, Gainesville, Florida 32610, United States

4. NEUROFARBA Department, Section of Pharmacology and Toxicology, University of Florence, Via G. Pieraccini 6, 50139 Florence, Italy

Funder

Universit?? degli Studi di Firenze

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01906

Reference46 articles.

1. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry

2. Structure-Based Design of Drugs and Other Bioactive Molecules

3. The development of drugs for treatment of sleeping sickness: a historical review

4. Triurea Derivatives of Diethylenetriamine as Potential Templates for the Formation of Artificial β-Sheets1

5. Solid-Phase Synthesis of Artificial β-Sheets

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