Design, Synthesis, and Biological Evaluation of New Type of Gemini Analogues with a Cyclopropane Moiety in Their Side Chain-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of New Type of Gemini Analogues with a Cyclopropane Moiety in Their Side Chain

Published:2024-06-10 Issue:12 Volume:67 Page:10386-10400
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gómez-Bouzó Uxía¹^ORCID,Peluso-Iltis Carole²³⁴⁵,Santalla Hugo¹,Quevedo Mario Alfredo⁶,Verlinden Lieve⁷^ORCID,Verstuyf Annemieke⁷,Fall Yagamare¹^ORCID,Gómez Generosa¹,Rochel Natacha²³⁴⁵^ORCID

Affiliation:

1. Departamento de Química Orgánica and Instituto de Investigación Sanitaría Galicia Sur (IISGS), Campus Lagoas Marcosende, Universidad de Vigo, Vigo 36310, Spain

2. Institute of Genetics and Molecular and Cellular Biology (IGBMC), Illkirch 67400, France

3. CNRS UMR 7104, Illkirch 67400, France

4. Inserm U1258, Illkirch 67400, France

5. University of Strasbourg, Illkirch 67400, France

6. Unidad de Investigación y desarrollo en Tecnología Farmacéutica (UNITEFA), CONICET and Departamento de Ciencias Farmacéuticas, Facultad de Ciencias Químicas, Universidad Nacional de Córdoba, Córdoba X5000HUA, Argentina

7. Clinical and Experimental Endocrinology, Department of Chronic Diseases and Metabolism, KU Leuven, Leuven 3000, Belgium

Funder

Agence Nationale de la Recherche

Fonds Wetenschappelijk Onderzoek

Xunta de Galicia

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.4c00854

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