Design, Synthesis, and Biological Evaluation of Small-Molecule-Based Radioligands with Improved Pharmacokinetic Properties for Imaging of Programmed Death Ligand 1-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of Small-Molecule-Based Radioligands with Improved Pharmacokinetic Properties for Imaging of Programmed Death Ligand 1

Published:2023-12-01 Issue:23 Volume:66 Page:15894-15915
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Krutzek Fabian¹,Donat Cornelius K.¹,Ullrich Martin¹,Stadlbauer Sven¹²^ORCID

Affiliation:

1. Helmholtz-Zentrum Dresden-Rossendorf, Institute of Radiopharmaceutical Cancer Research, Bautzner Landstraße 400, 01328 Dresden, Germany

2. Faculty of Chemistry and Food Chemistry, School of Science, Technische Universität Dresden, Mommsenstraße 4, 01069 Dresden, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c01355

Reference72 articles.

1. Efficacy of immune checkpoint inhibitor monotherapy for patients with massive non-small-cell lung cancer

2. Immune Checkpoint Inhibitors as Monotherapy or Within a Combinatorial Strategy in Advanced Hepatocellular Carcinoma

3. First-Line Immune-Checkpoint Inhibitors in Non-Small Cell Lung Cancer: Current Landscape and Future Progress

4. Development of Radiotracers for Imaging of the PD-1/PD-L1 Axis

5. PD-L1 Detection in Tumors Using [64Cu]Atezolizumab with PET

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Bioorthogonal Diels–Alder Click Chemistry-Based Pretargeted PET Imaging Strategy for Monitoring Programmed Death-Ligand 1 Expression;ACS Omega;2024-08-21

2. Application of 99mTc-Labeled WL12 Peptides as a Tumor PD-L1-Targeted SPECT Imaging Agent: Kit Formulation, Preclinical Evaluation, and Study on the Influence of Coligands;Pharmaceuticals;2024-07-08

3. Chelator impact: investigating the pharmacokinetic behavior of copper-64 labeled PD-L1 radioligands;EJNMMI Radiopharmacy and Chemistry;2024-02-19

4. Design, synthesis, and biological evaluation of a ^99mTc-labeled small-molecule tracer for PD-L1 imaging;New Journal of Chemistry;2024

5. Diagnostic and Therapeutic Radiopharmaceuticals: A “Hot” Topic;Journal of Medicinal Chemistry;2023-12-18