Lead Optimization of the 5-Phenylpyrazolopyrimidinone NPD-2975 toward Compounds with Improved Antitrypanosomal Efficacy-Reference-Cited by-同舟云学术

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Lead Optimization of the 5-Phenylpyrazolopyrimidinone NPD-2975 toward Compounds with Improved Antitrypanosomal Efficacy

Published:2024-02-08 Issue:4 Volume:67 Page:2849-2863
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zheng Yang¹^ORCID,van den Kerkhof Magali²,Ibrahim Mohamed¹,De Esch Iwan J. P.¹^ORCID,Maes Louis²,Sterk Geert Jan¹,Caljon Guy²,Leurs Rob¹^ORCID

Affiliation:

1. Amsterdam Institute of Molecular and Life Sciences, Division of Medicinal Chemistry, Faculty of Science, Vrije Universiteit Amsterdam, De Boelelaan 1108, Amsterdam 1081 HZ, The Netherlands

2. Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, Wilrijk 2610, Belgium

Funder

FP7 Health

China Scholarship Council

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c01976

Reference41 articles.

1. WHO. WHO HAT 2020, 2022. https://www.who.int/news-room/fact-sheets/detail/trypanosomiasis-human-african-(sleeping-sickness) (accessed 04 18, 2022).

2. Clinical and Neuropathogenetic Aspects of Human African Trypanosomiasis

3. Sleeping sickness: a tale of two diseases

4. The history of African trypanosomiasis

5. Human African trypanosomiasis

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1. An efficient One-Pot synthesis of NaOCl mediated pyrazolopyrimidine derivatives;Results in Chemistry;2024-10

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