Acetyl-Click Screening Platform Identifies Small-Molecule Inhibitors of Histone Acetyltransferase 1 (HAT1)-Reference-Cited by-同舟云学术

Acetyl-Click Screening Platform Identifies Small-Molecule Inhibitors of Histone Acetyltransferase 1 (HAT1)

Published:2023-04-07 Issue:8 Volume:66 Page:5774-5801
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gaddameedi Jitender D.¹,Chou Tristan²,Geller Benjamin S.²,Rangarajan Amithvikram²³,Swaminathan Tarun A.⁴,Dixon Danielle⁴,Long Katherine⁴^ORCID,Golder Caiden J.⁴^ORCID,Vuong Van A.⁴,Banuelos Selene²,Greenhouse Robert⁵,Snyder Michael P.²,Lipchik Andrew M.¹,Gruber Joshua J.⁴^ORCID

Affiliation:

1. Department of Pharmaceutical Sciences, Eugene Applebaum College of Pharmacy and Health Sciences, Wayne State University, Detroit, Michigan 48201, United States

2. Department of Genetics, Stanford University School of Medicine, Stanford, California 94309, United States

3. Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, California 94158, United States

4. Department of Internal Medicine, Hematology-Oncology Division, Cecil H. and Ida Green Center for Reproductive Biology Sciences, UT Southwestern Medical Center, Dallas, Texas 75235, United States

5. Department of Otolaryngology, Stanford University School of Medicine, Stanford, California 94309, United States

Funder

National Center for Advancing Translational Sciences

National Cancer Institute

National Human Genome Research Institute

National Institute of Diabetes and Digestive and Kidney Diseases

Basic Energy Sciences

Cancer Prevention and Research Institute of Texas

National Institute of General Medical Sciences

Stanford SPARK Scholars Award

Publisher

American Chemical Society (ACS)