Systematic Study of Heteroarene Stacking Using a Congeneric Set of Molecular Glues for Procaspase-6

Author:

Togo Takaya1,Tram Linh1,Denton Laura G.2,ElHilali-Pollard Xochina1,Gu Jun3,Jiang Jinglei3,Liu Chenglei3,Zhao Yan3,Zhao Yanlong3,Zheng Yinzhe3,Zheng Yunping3,Yang Jingjing3ORCID,Fan Panpan3,Arkin Michelle R.1ORCID,Härmä Harri4ORCID,Sun Deqian3,Canan Stacie S.5ORCID,Wheeler Steven E.2ORCID,Renslo Adam R.1ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, University of California, 600 16th Street, San Francisco, California 94143, United States

2. Department of Chemistry, University of Georgia, Athens, Georgia 30602, United States

3. Departments of Chemistry and Biology, Viva Biotech, Pu Dong New Area, 201203 Shanghai, China

4. Department of Chemistry, University of Turku, 20500 Turku, Finland

5. Departments of Chemistry and Structural Biology, Elgia Therapeutics, La Jolla, California 92037, United States

Funder

National Institute of General Medical Sciences

Merck

Uehara Memorial Foundation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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