Development of a New Class of CXCR4-Targeting Radioligands Based on the Endogenous Antagonist EPI-X4 for Oncological Applications

Author:

Gaonkar Raghuvir Haridas1ORCID,Schmidt Yannik Tim1,Mansi Rosalba1,Almeida-Hernandez Yasser23ORCID,Sanchez-Garcia Elsa23ORCID,Harms Mirja4,Münch Jan45ORCID,Fani Melpomeni1

Affiliation:

1. Division of Radiopharmaceutical Chemistry, Department Theragnostics, University Hospital Basel, Basel 4031, Switzerland

2. Computational Biochemistry, Center of Medical Biotechnology, University of Duisburg-Essen, Essen 45117, Germany

3. Computational Bioengineering, Faculty of Bio- and Chemical Engineering, Technical University Dortmund, Dortmund 44227, Germany

4. Institute of Molecular Virology, Ulm University Medical Center, Ulm 89081, Germany

5. Core Facility Functional Peptidomics, Ulm University Medical Center, Ulm 89081, Germany

Funder

Schweizerischer Nationalfonds zur Förderung der Wissenschaftlichen Forschung

Deutsche Forschungsgemeinschaft

Baden-Württemberg Stiftung

Universität Ulm

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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