Discovery of Nelutroctiv (CK-136), a Selective Cardiac Troponin Activator for the Treatment of Cardiovascular Diseases Associated with Reduced Cardiac Contractility
Author:
Affiliation:
1. Cytokinetics, Inc., 350 Oyster Point Boulevard, South San Francisco, California 94080, United States
Funder
Amgen
Cytokinetics
Publisher
American Chemical Society (ACS)
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c02413
Reference22 articles.
1. Cardiac Troponin Activator CK-963 Increases Cardiac Contractility in Rats
2. A Novel Small Molecule Troponin Activator Increases Cardiac Contractile Function Without Negative Impact on Energetics
3. Birth Prevalence of Congenital Heart Disease Worldwide
4. Systemic Right Ventricle in Adults With Congenital Heart Disease
5. Medical Therapy for Systemic Right Ventricles: A Systematic Review (Part 1) for the 2018 AHA/ACC Guideline for the Management of Adults With Congenital Heart Disease: A Report of the American College of Cardiology/American Heart Association Task Force on Clinical Practice Guidelines
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1. Maturation of human cardiac organoids enables complex disease modelling and drug discovery;2024-09-09
2. Cardiac Troponin Activator CK-963 Increases Cardiac Contractility in Rats;Journal of Medicinal Chemistry;2024-03-07
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