Celastrol Promotes Weight Loss in Diet-Induced Obesity by Inhibiting the Protein Tyrosine Phosphatases PTP1B and TCPTP in the Hypothalamus

Author:

Kyriakou Eleni12,Schmidt Stefanie12,Dodd Garron T.3,Pfuhlmann Katrin4567,Simonds Stephanie E.8,Lenhart Dominik129,Geerlof Arie1,Schriever Sonja C.457,De Angelis Meri10,Schramm Karl-Werner10,Plettenburg Oliver911ORCID,Cowley Michael A.8,Tiganis Tony312,Tschöp Matthias H.567,Pfluger Paul T.457,Sattler Michael12ORCID,Messias Ana C.12ORCID

Affiliation:

1. Institute of Structural Biology, Helmholtz Zentrum München, 85764 Neuherberg, Germany

2. Biomolecular NMR and Center for Integrated Protein Science Munich at Department of Chemistry, Technical University of Munich, 85747 Garching, Germany

3. Metabolism, Diabetes and Obesity Program, Biomedicine Discovery Institute, and Department of Biochemistry and Molecular Biology, Monash University, Victoria 3800, Australia

4. Research Unit Neurobiology of Diabetes, Helmholtz Zentrum München, 85764 Neuherberg, Germany

5. Institute for Diabetes and Obesity, Helmholtz Zentrum München, 85764 Neuherberg, Germany

6. Division of Metabolic Diseases, Technische Universität München, 80333 Munich, Germany

7. German Center for Diabetes Research (DZD), 85764 Neuherberg, Germany

8. Metabolism, Diabetes and Obesity Program, Biomedicine Discovery Institute, and Department of Physiology, Monash University, Victoria 3800, Australia

9. Institute of Medicinal Chemistry, Helmholtz Zentrum München, 85764 Neuherberg, Germany

10. Molecular EXposomics, Helmholtz Zentrum München, 85764 Neuherberg, Germany

11. Institute of Organic Chemistry, Leibniz Universität Hannover, 30167 Hannover, Germany

12. Peter MacCallum Cancer Centre, Melbourne, Victoria 3000, Australia

Funder

Helmholtz-Gemeinschaft

Department of Health, Australian Government

National Heart Foundation of Australia

Alexander von Humboldt-Stiftung

IMF Diabetes Portfolio Grant

Helmholtz-Israel-Cooperation in Personalized Medicine

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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