Design, (Radio)Synthesis, and in Vitro and in Vivo Evaluation of Highly Selective and Potent Matrix Metalloproteinase 12 (MMP-12) Inhibitors as Radiotracers for Positron Emission Tomography-Reference-Cited by-同舟云学术

Design, (Radio)Synthesis, and in Vitro and in Vivo Evaluation of Highly Selective and Potent Matrix Metalloproteinase 12 (MMP-12) Inhibitors as Radiotracers for Positron Emission Tomography

Published:2018-04-16 Issue:9 Volume:61 Page:4115-4134
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Butsch Viktoria¹,Börgel Frederik²,Galla Fabian²,Schwegmann Katrin³,Hermann Sven³,Schäfers Michael¹³⁴,Riemann Burkhard¹,Wünsch Bernhard²⁴,Wagner Stefan¹^ORCID

Affiliation:

1. Department of Nuclear Medicine, University Hospital Münster, Albert-Schweitzer-Campus 1, Building A1, 48149 Münster, Germany

2. Institute of Pharmaceutical and Medicinal Chemistry, University of Münster, Corrensstraße 48, 48149 Münster, Germany

3. European Institute for Molecular Imaging, University of Münster, Waldeyerstraße 15, 48149 Münster, Germany

4. Cells-in-Motion Cluster of Excellence (EXC 1003 − CiM), University of Münster, 48149 Münster, Germany

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b00200

Reference65 articles.

1. Structural Basis of Matrix Metalloproteinases and Tissue Inhibitors of Metalloproteinases

2. Intricate Functions of Matrix Metalloproteinases in Physiological and Pathological Conditions

3. Matrix Metalloproteinases in Non-Neoplastic Disorders

4. Matrix metalloproteinases (MMPs), the main extracellular matrix (ECM) enzymes in collagen degradation, as a target for anticancer drugs

5. Targeting matrix metalloproteinases in cancer: Bringing new life to old ideas

Cited by 37 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Organocatalytic route to the enantioselective synthesis of syn/anti-α-hydrazino-γ-fluoro alcohols;Tetrahedron Letters;2024-07

2. Organocatalytic Route to the Enantioselective Synthesis of Syn/Anti-Α-Hydrazino-ℽ-Fluoro Alcohols;2024

3. Transition Metal-catalyzed Regioselective Direct C-H Arylations Using Quinone Diazide as Arylating Agent: A Mini Review;Mini-Reviews in Organic Chemistry;2023-08

4. Matrix Metalloproteinases Inhibitors in Cancer Treatment: An Updated Review (2013–2023);Molecules;2023-07-21

5. Conformationally Restricted?1 Receptor Antagonists from (-)-Isopulegol;J MED CHEM;2023