Pyrrolone Derivatives as Intracellular Allosteric Modulators for Chemokine Receptors: Selective and Dual-Targeting Inhibitors of CC Chemokine Receptors 1 and 2
Author:
Affiliation:
1. Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands
Funder
Agentschap Innoveren en Ondernemen
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b00605
Reference67 articles.
1. Chemokines and Chemokine Receptors: Positioning Cells for Host Defense and Immunity
2. International Union of Basic and Clinical Pharmacology. LXXXIX. Update on the Extended Family of Chemokine Receptors and Introducing a New Nomenclature for Atypical Chemokine Receptors
3. New paradigms in chemokine receptor signal transduction: Moving beyond the two-site model
4. Chemokines and their receptors: insights from molecular modeling and crystallography
5. Beyond Chemoattraction: Multifunctionality of Chemokine Receptors in Leukocytes
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