Boron-Pleuromutilins as Anti-Wolbachia Agents with Potential for Treatment of Onchocerciasis and Lymphatic Filariasis

Author:

Jacobs Robert T.1ORCID,Lunde Christopher S.1,Freund Yvonne R.1,Hernandez Vincent1,Li Xianfeng1,Xia Yi1,Carter David S.1,Berry Pamela W.1,Halladay Jason1,Rock Fernando1,Stefanakis Rianna1,Easom Eric1,Plattner Jacob J.1,Ford Louise2,Johnston Kelly L.2,Cook Darren A. N.2,Clare Rachel2,Cassidy Andrew2,Myhill Laura2,Tyrer Hayley2,Gamble Joanne2,Guimaraes Ana F.2,Steven Andrew2,Lenz Franziska3,Ehrens Alexandra3,Frohberger Stefan J.3,Koschel Marianne3,Hoerauf Achim3,Hübner Marc P.3,McNamara Case W.4,Bakowski Malina A.4,Turner Joseph D.2,Taylor Mark J.2,Ward Stephen A.2

Affiliation:

1. Anacor Pharmaceuticals, 1020 East Meadow Circle, Palo Alto, California 94303, United States

2. Centre for Drugs and Diagnostics, Department of Parasitology, Liverpool School of Tropical Medicine, Pembroke Place, Liverpool L3 5QA, U.K.

3. Institute for Medical Microbiology, Immunology and Parasitology, University Hospital Bonn, Sigmund Freud Str. 25, 53127 Bonn, Germany

4. Calibr, 11119 North Torrey Pines Road, Suite 100, La Jolla, California 92037, United States

Funder

Bill and Melinda Gates Foundation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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