Potent Metabolic Sialylation Inhibitors Based on C-5-Modified Fluorinated Sialic Acids

Author:

Heise Torben1,Pijnenborg Johan F. A.1,Büll Christian2,van Hilten Niek3,Kers-Rebel Esther D.2,Balneger Natasja2,Elferink Hidde1,Adema Gosse J.2,Boltje Thomas J.1ORCID

Affiliation:

1. Cluster for Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525AJ, The Netherlands

2. Radiotherapy & OncoImmunology Laboratory, Department of Radiation Oncology, Radboudumc, Nijmegen 6525 GA, The Netherlands

3. Supramolecular and Biomaterials Chemistry, Leiden Institute of Chemistry, Leiden University, Leiden 2333 CC, The Netherlands

Funder

H2020 European Research Council

KWF Kankerbestrijding

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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