Molecular Basis for the N-Terminal Bromodomain-and-Extra-Terminal-Family Selectivity of a Dual Kinase–Bromodomain Inhibitor-Reference-Cited by-同舟云学术

Molecular Basis for the N-Terminal Bromodomain-and-Extra-Terminal-Family Selectivity of a Dual Kinase–Bromodomain Inhibitor

Published:2018-09-25 Issue:20 Volume:61 Page:9316-9334
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Divakaran Anand¹^ORCID,Talluri Siva K.²,Ayoub Alex M.²,Mishra Neeraj K.²,Cui Huarui²,Widen John C.¹,Berndt Norbert³,Zhu Jin-Yi³,Carlson Angela S.²,Topczewski Joseph J.²^ORCID,Schonbrunn Ernst K.³^ORCID,Harki Daniel A.¹^ORCID,Pomerantz William C. K.¹²^ORCID

Affiliation:

1. Department of Medicinal Chemistry, University of Minnesota, 2231 6th Street SE, Minneapolis, Minnesota 55455, United States

2. Department of Chemistry, University of Minnesota, 207 Pleasant Street SE, Minneapolis, Minnesota 55455, United States

3. Drug Discovery Department, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States

Funder

Division of Chemistry

National Cancer Institute

American Heart Association

National Institute of General Medical Sciences

Masonic Cancer Center, University of Minnesota

Publisher

American Chemical Society (ACS)