Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach-Reference-Cited by-同舟云学术

Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach

Published:2017-11-20 Issue:24 Volume:60 Page:10013-10025
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Anumala Upendra Rao¹,Waaler Jo²³,Nkizinkiko Yves⁴,Ignatev Alexander⁴,Lazarow Katina¹,Lindemann Peter¹,Olsen Petter Angell²³,Murthy Sudarshan⁴,Obaji Ezeogo⁴,Majouga Alexander G.⁵,Leonov Sergey⁶⁷,von Kries Jens Peter¹⁸,Lehtiö Lari⁴^ORCID,Krauss Stefan²³,Nazaré Marc¹⁸^ORCID

Affiliation:

1. Leibniz-Forschungsinstitut für Molekulare Pharmakologie (FMP), Campus Berlin-Buch, 13125 Berlin, Germany

2. Unit for Cell Signaling, Institute of Medical Microbiology, Oslo University Hospital, Gaustadalleen 34, 0372 Oslo, Norway

3. Hybrid Technology Hub, Centre of Excellence, Institute of Basic Medical Sciences, University of Oslo, 0372 Oslo, Norway

4. Faculty of Biochemistry and Molecular Medicine, Biocenter Oulu, University of Oulu, P.O. Box 5400, 90014 Oulu, Finland

5. Department of Chemistry, Moscow State University, Leninskie Gory 1/3, Moscow 119991, Russia

6. National University of Science and Technology MISiS, Leninsky Avenue 4, Moscow 119049, Russia

7. Moscow Institute of Physics and Technology (State University), Institutskiy Lane 9, 141700 Dolgoprudny, Russia

8. Berlin Institute of Health (BIH), Anna-Louisa-Karsch-Strasse 2, 10178 Berlin, Germany

Funder

Sigrid Jus?liuksen S??ti?

Norges Forskningsr?d

Jane ja Aatos Erkon S??ti?

Suomen Akatemia

Ministry of Education and Science of the Russian Federation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00883

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