Development of (4-Cyanophenyl)glycine Derivatives as Reversible Inhibitors of Lysine Specific Demethylase 1-Reference-Cited by-同舟云学术

Development of (4-Cyanophenyl)glycine Derivatives as Reversible Inhibitors of Lysine Specific Demethylase 1

Published:2017-09-21 Issue:19 Volume:60 Page:7984-7999
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mould Daniel P.¹^ORCID,Alli Cristina²,Bremberg Ulf³,Cartic Sharon²,Jordan Allan M.¹^ORCID,Geitmann Matthis³,Maiques-Diaz Alba⁴,McGonagle Alison E.¹,Somervaille Tim C. P.⁴,Spencer Gary J.⁴,Turlais Fabrice²,Ogilvie Donald¹

Affiliation:

1. Drug Discovery Unit, Cancer Research UK Manchester Institute, University of Manchester, Wilmslow Road, Manchester, M20 4BX, U.K.

2. CRT Discovery Laboratories, Babraham Campus, Babraham, Cambridgeshire CB22 3AT, U.K.

3. Beactica AB, Uppsala Business Park, Virdings allé 2, 75450, Uppsala, Sweden

4. Leukaemia Biology Laboratory, Cancer Research UK Manchester Institute, University of Manchester, Wilmslow Road, Manchester, M20 4BX, U.K.

Funder

Cancer Research UK

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00462

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