Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors-Reference-Cited by-同舟云学术

Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors

Published:2017-11-22 Issue:23 Volume:60 Page:9790-9806
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bayliss Tracy¹,Robinson David A.¹^ORCID,Smith Victoria C.¹,Brand Stephen¹,McElroy Stuart P.¹,Torrie Leah S.¹,Mpamhanga Chido¹,Norval Suzanne¹,Stojanovski Laste¹,Brenk Ruth¹,Frearson Julie A.¹,Read Kevin D.¹,Gilbert Ian H.¹^ORCID,Wyatt Paul G.¹^ORCID

Affiliation:

1. Drug Discovery Unit, College of Life Sciences, University of Dundee, Sir James Black Centre, Dundee DD1 5EH, U.K.

Funder

Wellcome Trust

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01255

Reference45 articles.

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4. The continuing problem of human African trypanosomiasis (sleeping sickness)

5. Drug used in the treatment of sleeping sickness (human African trypanosomiasis: HAT)

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