A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors-Reference-Cited by-同舟云学术

A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors

Published:2017-12-11 Issue:24 Volume:60 Page:10151-10171
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bronner Sarah M.¹^ORCID,Murray Jeremy¹,Romero F. Anthony¹^ORCID,Lai Kwong Wah²,Tsui Vickie¹,Cyr Patrick¹^ORCID,Beresini Maureen H.¹,de leon Boenig Gladys¹,Chen Zhongguo²,Choo Edna F.¹^ORCID,Clark Kevin R.¹,Crawford Terry D.¹^ORCID,Jayaram Hariharan³,Kaufman Susan¹,Li Ruina¹,Li Yingjie²,Liao Jiangpeng²,Liang Xiaorong¹,Liu Wenfeng²,Ly Justin¹,Maher Jonathan¹,Wai John²,Wang Fei²,Zheng Aijun²,Zhu Xiaoyu²,Magnuson Steven¹

Affiliation:

1. Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States

2. Wuxi Apptec Co., Ltd., 288 Fute Zhong Road, Waigaoqiao Free Trade Zone, Shanghai 200131, People’s Republic of China

3. Editas Medicine, Inc., 11 Hurley Street, Cambridge, Massachusetts 02141, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01372

Reference60 articles.

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