Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity-Reference-Cited by-同舟云学术

Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity

Published:2017-10-16 Issue:20 Volume:60 Page:8647-8660
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

dos Santos Fernandes Guilherme Felipe¹²³^ORCID,de Souza Paula Carolina²⁴,Moreno-Viguri Elsa³^ORCID,Santivañez-Veliz Mery³,Paucar Rocio³,Pérez-Silanes Silvia³^ORCID,Chegaev Konstantin⁵^ORCID,Guglielmo Stefano⁵^ORCID,Lazzarato Loretta⁵^ORCID,Fruttero Roberta⁵,Man Chin Chung²,da Silva Patricia Bento²,Chorilli Marlus²^ORCID,Solcia Mariana Cristina²,Ribeiro Camila Maríngolo²,Silva Caio Sander Paiva²,Marino Leonardo Biancolino²,Bosquesi Priscila Longhin²,Hunt Debbie M.⁶,de Carvalho Luiz Pedro S.⁶,de Souza Costa Carlos Alberto⁷,Cho Sang Hyun⁴,Wang Yuehong⁴,Franzblau Scott Gary⁴,Pavan Fernando Rogério²,dos Santos Jean Leandro¹²^ORCID

Affiliation:

1. São Paulo State University (UNESP), Institute of Chemistry, Araraquara 14800060, Brazil

2. São Paulo State University (UNESP), School of Pharmaceutical Sciences, Araraquara 14800903, Brazil

3. Universidad de Navarra, Department of Organic and Pharmaceutical Chemistry, Instituto de Salud Tropical, Pamplona 31008, Spain

4. Institute of Tuberculosis Research, University of Illinois at Chicago, Chicago, Illinois 60607, United States

5. Dipartimento di Scienza e Tecnologia del Farmaco, Università degli Studi di Torino, Turin 10124, Italy

6. Mycobacterial Metabolism and Antibiotic Research Laboratory, The Francis Crick Institute, 1 Midland Road, London NW1 1AT, United Kingdom

7. São Paulo State University (UNESP), School of Odontology, Araraquara 14801903, Brazil

Funder

Medical Research Council

National Institute of Allergy and Infectious Diseases

Conselho Nacional de Desenvolvimento Cient?fico e Tecnol?gico

Wellcome Trust

Funda??o de Amparo ? Pesquisa do Estado de S?o Paulo

Cancer Research UK

Pr?-Reitoria de P?s-Gradua??o, Universidade Estadual Paulista

Faculdade de Ci?ncias Farmac?uticas, Universidade Estadual Paulista "J?lio de Mesquita Filho"

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01332

Reference74 articles.

1. Global Tuberculosis Report 2016;World Health Organization:Geneva, Switzerland, 2016.

2. Global Tuberculosis Report 2013;World Health Organization:Geneva, Switzerland, 2013.

3. The Enduring Hypoxic Response of Mycobacterium tuberculosis

4. Models of Latent Tuberculosis: Their Salient Features, Limitations, and Development

5. Advances in the development of new tuberculosis drugs and treatment regimens

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