Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists-Reference-Cited by-同舟云学术

Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists

Published:2017-10-24 Issue:21 Volume:60 Page:8716-8730
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Palmer Daniel¹^ORCID,Gonçalves Juliana P. L.¹^ORCID,V. Hansen Louise¹,Wu Boqian²,Hald Helle¹,Schoffelen Sanne¹,Diness Frederik¹,Le Quement Sebastian T.³,Nielsen Thomas E.⁴⁵⁶,Meldal Morten¹

Affiliation:

1. CECB, Department of Chemistry, University of Copenhagen, Universitetsparken 5, 2100 Copenhagen, Denmark

2. Aquaporin A/S, Ole Maaløes Vej 3, 2200 Copenhagen, Denmark

3. CMC API Development, Novo Nordisk A/S, Novo Nordisk Park, 2760 Måløv, Denmark

4. Protein & Peptide Chemistry, Novo Nordisk A/S, Novo Nordisk Park, 2760 Måløv, Denmark

5. Department of Immunology and Microbiology, University of Copenhagen, Blegdamsvej 3B, 2200 Copenhagen, Denmark

6. Singapore Centre on Environmental Life Sciences Engineering, Nanyang Technological University, 60 Nanyang Drive, SG 637551, Singapore

Funder

Danmarks Grundforskningsfond

K?benhavns Universitet

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00353

Reference90 articles.

1. Are GPCRs Still a Source of New Targets?

2. Comprehensive repertoire and phylogenetic analysis of the G protein-coupled receptors in human and mouse

3. The GRAFS classification system of G-protein coupled receptors in comparative perspective

4. 60 YEARS OF POMC: Melanocortin receptors: evolution of ligand selectivity for melanocortin peptides

5. MOLECULAR EVOLUTION OF GPCRS: Melanocortin/melanocortin receptors

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