Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors-Reference-Cited by-同舟云学术

Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors

Published:2018-03-28 Issue:8 Volume:61 Page:3454-3477
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sellmer Andreas¹,Stangl Hubert²,Beyer Mandy³,Grünstein Elisabeth¹,Leonhardt Michel¹,Pongratz Herwig¹,Eichhorn Emerich¹,Elz Sigurd¹,Striegl Birgit⁴⁵,Jenei-Lanzl Zsuzsa²⁶,Dove Stefan¹,Straub Rainer H.²,Krämer Oliver H.³,Mahboobi Siavosh¹^ORCID

Affiliation:

1. Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, 93040 Regensburg, Germany

2. Laboratory of Experimental Rheumatology and Neuroendocrine Immunology, Department of Internal Medicine, University Hospital, 93042 Regensburg, Germany

3. Institute of Toxicology, University Medical Center Mainz, 55131 Mainz, Germany

4. Technical University of Applied Sciences (OTH) Regensburg, 93053 Regensburg, Germany

5. Regensburg Center of Biomedical Engineering (RCBE), OTH and University Regensburg, 93053 Regensburg, Germany

6. Dr. Rolf M. Schwiete Research Unit for Osteoarthritis, Orthopedic University Hospital, Friedrichsheim gGmbH, 60528 Frankfurt/Main, Germany

Funder

Deutsche Forschungsgemeinschaft

Wilhelm Sander-Stiftung

Deutsche Krebshilfe

Naturwissenschaftlich-medizinisches Forschungszentrum, Johannes Gutenberg-Universit?t

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01593

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