Synthesis and Structure–Activity Relationships of the Novel Antimalarials 5-Pyridinyl-4(1H)-Pyridones-Reference-Cited by-同舟云学术

Synthesis and Structure–Activity Relationships of the Novel Antimalarials 5-Pyridinyl-4(1H)-Pyridones

Published:2018-03-28 Issue:8 Volume:61 Page:3422-3435
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bueno José M.¹,Calderon Félix¹^ORCID,Chicharro Jesús¹,De la Rosa Juan C.¹,Díaz Beatriz¹,Fernández Jorge¹,Fiandor José M.¹,Fraile María T.¹,García Mercedes¹,Herreros Esperanza¹,García-Pérez Adolfo¹,Lorenzo Milagros¹,Mallo Araceli¹^ORCID,Puente Margarita¹,Saadeddin Anas¹,Ferrer Santiago¹,Angulo-Barturen Iñigo¹,Burrows Jeremy N.²,León María L.¹^ORCID

Affiliation:

1. Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Calle de Severo Ochoa, 2, 28760 Tres Cantos, Madrid, Spain

2. Medicines for Malaria Venture, ICC, Route de Pré-Bois 20, PO Box 1826, 1215 Geneva, Switzerland

Funder

Medicines for Malaria Venture

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01256

Reference42 articles.

1. World malaria report 2016; World Health Organization: Geneva, Switzerland, 2016. Available at http://www.who.int/malaria/publications/world-malaria-report-2016/report/en/.

2. The Global Portfolio of New Antimalarial Medicines Under Development

3. The clinical impact of artemisinin resistance in Southeast Asia and the potential for future spread

4. Antimalarial drug resistance: linking Plasmodium falciparum parasite biology to the clinic

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