Discovery of Potent and Brain-Penetrant GPR52 Agonist that Suppresses Psychostimulant Behavior-Reference-Cited by-同舟云学术

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Discovery of Potent and Brain-Penetrant GPR52 Agonist that Suppresses Psychostimulant Behavior

Published:2020-11-16 Issue:22 Volume:63 Page:13951-13972
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wang Pingyuan¹,Felsing Daniel E.²,Chen Haiying¹,Stutz Sonja J.²,Murphy Ryan E.²,Cunningham Kathryn A.¹²^ORCID,Allen John A.¹²,Zhou Jia¹²^ORCID

Affiliation:

1. Chemical Biology Program, Department of Pharmacology and Toxicology, University of Texas Medical Branch, Galveston, Texas 77555, United States

2. Center for Addiction Research, University of Texas Medical Branch, Galveston, Texas 77555, United States

Funder

National Institute on Drug Abuse

Pharmaceutical Research and Manufacturers of America Foundation

University of Texas Medical Branch

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01498

Reference35 articles.

1. Strategies to Discover Unexpected Targets for Drugs Active at G Protein–Coupled Receptors

2. Allosteric Modulation of Class A GPCRs: Targets, Agents, and Emerging Concepts

3. GPCR Drug Discovery: Emerging Targets, Novel Approaches and Future Trends

4. How many drug targets are there?

5. Structural diversity of G protein-coupled receptors and significance for drug discovery

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2. Exploring orphan GPCRs in neurodegenerative diseases;Frontiers in Pharmacology;2024-06-04

3. Discovery of 3-((4-Benzylpyridin-2-yl)amino)benzamides as Potent GPR52 G Protein-Biased Agonists;Journal of Medicinal Chemistry;2024-05-24

4. Orphan GPR52 as an emerging neurotherapeutic target;Drug Discovery Today;2024-04

5. The non-nutritive sweetener sucralose increases β-arrestin signaling at the constitutively active orphan G protein-coupled receptor GPR52;Canadian Journal of Physiology and Pharmacology;2024-02-01

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