Discovery of Potent and Selective PI3Kγ Inhibitors
Author:
Affiliation:
1. Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01203
Reference29 articles.
1. PI3K-AKT-mTOR inhibition in cancer immunotherapy, redux
2. PI3K in cancer: divergent roles of isoforms, modes of activation and therapeutic targeting
3. Targeting PI3K in cancer: mechanisms and advances in clinical trials
4. The Hallmarks of Cancer
5. Hallmarks of Cancer: The Next Generation
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