Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2-Reference-Cited by-同舟云学术

Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2

Published:2020-06-26 Issue:14 Volume:63 Page:7766-7772
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lindenblatt Dirk¹^ORCID,Nickelsen Anna²^ORCID,Applegate Violetta M.¹^ORCID,Jose Joachim²^ORCID,Niefind Karsten¹^ORCID

Affiliation:

1. Department für Chemie, Institut für Biochemie, Universität zu Köln, Zülpicher Str. 47, D-50674 Köln, Germany

2. Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität Münster, PharmaCampus, Corrensstr. 48, D-48149 Münster, Germany

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00587

Reference48 articles.

1. The Evolution of Protein Kinase Inhibitors from Antagonists to Agonists of Cellular Signaling

2. New Directions in Targeting Protein Kinases: Focusing Upon True Allosteric and Bivalent Inhibitors

3. Protein kinase CK2: structure, regulation and role in cellular decisions of life and death

4. Crystal structure of human protein kinase CK2: insights into basic properties of the CK2 holoenzyme

5. Protein Kinase CK2 in Human Diseases

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