Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D-Reference-Cited by-同舟云学术

Structure–Activity Relationship Studies of Pyrimidine-4-Carboxamides as Inhibitors of N-Acylphosphatidylethanolamine Phospholipase D

Published:2020-12-31 Issue:1 Volume:64 Page:481-515
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mock Elliot D.¹^ORCID,Kotsogianni Ioli¹,Driever Wouter P. F.¹,Fonseca Carmen S.¹,Vooijs Jelle M.¹,den Dulk Hans¹,van Boeckel Constant A. A.¹,van der Stelt Mario¹

Affiliation:

1. Department of Molecular Physiology, Leiden Institute of Chemistry, Leiden University and Oncode Institute, 2300 RA Leiden, Netherlands

Funder

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Faculty of Science, Leiden University

Oncode Institute

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01441

Reference22 articles.

1. Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

2. Molecular Characterization of a Phospholipase D Generating Anandamide and Its Congeners

3. Endocannabinoids and related N-acylethanolamines: biological activities and metabolism

4. Metabolism of the Endocannabinoid Anandamide: Open Questions after 25 Years

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