Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site-Reference-Cited by-同舟云学术

Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site

Published:2021-04-27 Issue:9 Volume:64 Page:5766-5786
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Knox Alexandra K.¹,Kalchschmid Christina¹,Schuster Daniela¹²^ORCID,Gaggia Francesca¹,Gust Ronald¹^ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, Institute of Pharmacy, CMBI − Center for Molecular Biosciences Innsbruck, University of Innsbruck, CCB − Center for Chemistry and Biomedicine, 6020 Innsbruck, Austria

2. Department of Pharmaceutical and Medicinal Chemistry, Institute of Pharmacy, Paracelsus Medical University, 5020 Salzburg, Austria

Funder

?sterreichische Forschungsf?rderungsgesellschaft

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c02230

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1. Global, Regional, and National Cancer Incidence, Mortality, Years of Life Lost, Years Lived With Disability, and Disability-Adjusted Life-Years for 29 Cancer Groups, 1990 to 2017

2. Breast Cancer, Estrogen Receptor and Ligands

3. Selective Estrogen-Receptor Modulators and Antihormonal Resistance in Breast Cancer

4. Biological determinants of endocrine resistance in breast cancer

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