CC-90009: A Cereblon E3 Ligase Modulating Drug That Promotes Selective Degradation of GSPT1 for the Treatment of Acute Myeloid Leukemia-Reference-Cited by-同舟云学术

CC-90009: A Cereblon E3 Ligase Modulating Drug That Promotes Selective Degradation of GSPT1 for the Treatment of Acute Myeloid Leukemia

Published:2021-02-16 Issue:4 Volume:64 Page:1835-1843
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hansen Joshua D.¹^ORCID,Correa Matthew¹,Alexander Matt¹,Nagy Mark¹,Huang Dehua¹,Sapienza John¹,Lu Gang¹,LeBrun Laurie A.¹,Cathers Brian E.¹,Zhang Weihong²,Tang Yang¹,Ammirante Massimo¹,Narla Rama K.¹,Piccotti Joseph R.¹,Pourdehnad Michael³,Lopez-Girona Antonia¹

Affiliation:

1. Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States

2. Bristol Myers Squibb, 556 Morris Avenue, Summit, New Jersey 07901, United States

3. Bristol Myers Squibb, 1500 Owens Street, Suite 600, San Francisco, California 94158, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01489

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