N-Trifluoromethyl Amines and Azoles: An Underexplored Functional Group in the Medicinal Chemist’s Toolbox-Reference-Cited by-同舟云学术

N-Trifluoromethyl Amines and Azoles: An Underexplored Functional Group in the Medicinal Chemist’s Toolbox

Published:2020-10-28 Issue:21 Volume:63 Page:13076-13089
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Schiesser Stefan¹^ORCID,Chepliaka Hanna¹²,Kollback Johanna¹³,Quennesson Thibaut¹⁴,Czechtizky Werngard¹,Cox Rhona J.¹

Affiliation:

1. Department of Medicinal Chemistry, Research and Early Development, Respiratory & Immunology, BioPharmaceuticals R&D, AstraZeneca, Pepparedsleden 1, 43183 Mölndal, Sweden

2. Department of Chemistry, Ludwig-Maximilians Universität München, Butenandstrasse 5−13, 81377 Munich, Germany

3. Department of Chemistry and Molecular Biology, Göteborgs universitet, Kemigården 4, 41296 Gothenburg, Sweden

4. Université de Lille, Institut Pasteur de Lille, INSERM U1177 − Drugs and Molecules for Living Systems, 59000 Lille, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01457

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