Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure–Activity Relationship Studies

Author:

Gonzalez Simon1,Dumitrascuta Maria2,Eiselt Emilie3,Louis Stevany2,Kunze Linda2,Blasiol Annalisa2,Vivancos Mélanie3,Previti Santo1,Dewolf Elke1,Martin Charlotte1,Tourwé Dirk1,Cavelier Florine4ORCID,Gendron Louis3ORCID,Sarret Philippe3ORCID,Spetea Mariana2ORCID,Ballet Steven1ORCID

Affiliation:

1. Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium

2. Department of Pharmaceutical Chemistry, Institute of Pharmacy and Center for Molecular Biosciences Innsbruck (CMBI), University of Innsbruck, 6020 Innsbruck, Austria

3. Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, J1H 5N4 Sherbrooke, Canada

4. Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, 34095 Montpellier, France

Funder

Canadian Institutes of Health Research

Fonds de Recherche du Qu?bec - Sant?

Universit?t Innsbruck

Austrian Science Fund

Canada Research Chairs

Fonds Wetenschappelijk Onderzoek

Natural Sciences and Engineering Research Council of Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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